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Raw Tianeptine hemisulfate monohydrate hmoov (1224690-84-9)

nyob 5.00 tawm ntawm 5 raws li nyob rau hauv 1 neeg ntsuam xyuas
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Tianeptine Sulfate, tseem hu ua Raw Tianeptine hemisulfate monohydrate hmoov, yog ib qho ......


raws li txoj cai: Hauv Pawg Ntau Lawm
Chav: 25kg / Nruas
Peev Xwm: 1350kg / hli

Hauj lwm

Raw Tianeptine hemisulfate monohydrate hmoov (1224690-84-9) video

Raw Tianeptine hemisulfate monohydrate hmoov (1224690-84-9) Specifications

khoom npe Raw Tianeptine hemisulfate monohydrate hmoov
Tshuaj Npe Tshuaj Tianeptine hemisulfate monohydrate; 1224690-84-9; Heptanoic acid,
Hom NAme Stablon, Coaxil
Chav Kawm Tshuaj Intermediates & Fine Tshuaj
CAS Number 1224690-84-9
Hauv Chikey KVVMXNNJBVTOSX-UHFFFAOYSA-N
molecular Formula C42H56Cl2N4O14S3
molecular Wyim 1008.004 g / mol
Monoisotopic pawg 1006.233 g / mol
Melting Point 1800 ℃
Kub npau npau Point 269.8 ° C ntawm 760 mmHg
Loj Ib Nrab Ntawm Ib Leeg N / A
xim so-dawb hmoov
Solubility Freetly soluble Nyob hauv dej thiab methanol thiab dichloromethane
Snkauj Thuab cua Txias qhuav qhov chaw
Application Tianeptine sodium tuaj yeem siv hauv Tricyclic compound nrog kev puas hlwb

Tianeptine sodium muaj nuj nqi kev tiv thaiv kab mob thiab kev tiv thaiv tsis tau cov khoom. Antidepressant

Raw Tianeptine hemisulfate monohydrate (THM) hmoov (1224690-84-9)

Raw Tianeptine hemisulfate monohydrate hmoov, kuj hu ua Tianeptine Sulfate, yog ib qho kev txhim kho version ntawm tianeptine sodium ntsev daim ntawv. Nws tsis yog-hygroscopic, yooj yim lis, mus yoo yooj yim dua, thiab kav ntev li ob zaug. Nws muaj tag nrho cov txiaj ntsim zoo tib yam li Tianeptine Sodium, tsuas yog daim ntawv sulfate muaj ib nrab hnub ntawm 5-6 cov xuab moos, yog li nws yuav kav ntev li ntev li ntev li tianeptine sodium. Vim li no, cov kws tshawb fawb yuav tsum xav tau 2-3 lub sij hawm cov dej sulfate kom ua tiav cov kev xav tau uas lawv tau tuaj yeem los ntawm sodium. Sulfate tseem muaj tsawg heev nyob rau hauv ob qho tib si saj thiab viscosity.

Tianeptine hemisulfate monohydrate yog cais raws li xim serotonin reuptake enhancer (SSRE) siv los kho kev nyuaj siab. Tianeptine tau tsim nyob rau hauv Fabkis nyob rau hauv 1960s thiab tau siv thoob plaws hauv lub xeem ib feem ntawm 2000s.

Nws kuj tseem siv tau los kho mob siab plob tsis so tswj siab lossis mob hawb pob. Thaum hnyav koob nws tau tshaj tawm los tsim cov kev ua si zoo li opioid xws li sedation thiab stimulation, motivation li, thiab euphoria thaum muab.

Tianeptine hemisulfate monohydrate (THM) hmoov (1224690-84-9) Mechanism of Action

Ib hom kev ua yeeb yam rau Tianeptine hemisulfate monohydrate yog kom nce siab rau serotonin (5-HT) hauv lub paj hlwb thiab hauv platelets. Tsis zoo li feem ntau cov khoos kas tricyclic, Tianeptine tsis tuaj yeem tshwm sim nrog kev ua rau lub peev xwm los sis lub cev muaj zog. Nws zoo nkaus li muaj kev ua si ntawm glutamatergic system, uas yog hypothesized los ua ib tug tshiab antidepressant mechanism.

Los ntawm kev ua kom cov nquab tuaj txog serotonin, Tianeptine hemisulfate monohydrate muaj ib cov lus sib txawv rau cov tshuaj SSRIs. Tsis ntev los no cov kev tshawb fawb tau soj ntsuam cov teebmeem ntawm Tianeptine hauv lub moj khaum ntawm qhov kev xav ntawm kev nyuaj siab, uas nws muaj qee yam kev ua. Tsis ntev los no cov kev tshawb fawb tseem qhia tau tias Tianeptine yuav muaj kev sib raug zoo nrog adenosine A1 tus neeg tau txais kev pab (receptors).

Tsis tas li ntawd, kev tshawb fawb tsis ntev los no luam tawm hauv 2014 qhia tias Tianeptine yuav ua tau raws li tus kab mob hu ua m -opioid receptor (MOR) agonist. Cov neeg tshawb nrhiav siv radioligand dabtsi thiab kev sib tw ntawm tes los soj ntsuam Tianeptine ua ib qho zoo MOR agonist. Nws kuj yog ib qho kev d-opioid agonist tab sis ntawm qis dua qis heev. Tianeptine tsis muaj nyob hauv k-opioid receptor chaw.

siv ntawm Tianeptine hemisulfate monohydrate (THM) hmoov (1224690-84-9)

▪ Kev nyuaj siab heev

▪ Cov kev ntxhov siab thiab kev ntxub ntxaug thiab cov tshuaj tsis zoo

▪ Kev paub kev txawj ntse thiab kev kawm zoo tuaj

▪ Mob leeg

▪ ADHD

Pom zoo Tianeptine hemisulfate monohydrate (THM) hmoov (1224690-84-9)

Tianeptine hemisulfate monohydrate tsuas yog 25 mg ib zaug, lossis ob zaug ib hnub. Txawm tias thaum pib nrog cov tshuaj tsis muaj zog, nws zoo tshaj rau kev txwv rau 2 lossis 3 hnub ib lub lim tiam nrog tsawg kawg ntawm 3 - 4 hnub hauv nruab nrab.

Tianeptine hemisulfate monohydrate los hauv daim ntawv tshuaj los yog hmoov. Nws raug nquahu kom pib nrog kev noj tshuaj tsawg thiab nce ntxiv tsawg txog rau cov tshuaj npaum li cas. Tsis tas li xwb, koob tshuaj me me ua rau kom muaj kev quav yeeb quav tshuaj, hnyav heev, thiab ua siab ntev.

Kab mob ntawm 50 - 75 mg yuav ua rau kev mob nkeeg. Tus Tianeptine hemisulfate monohydrate ua si ntawm> 100 mg yuav ua rau Tianeptine hemisulfate monohydrate siab.

Cov txiaj ntsig ntawm Tianeptine hemisulfate monohydrate (THM) hmoov (1224690-84-9)

♦ Tianeptine hemisulfate monohydrate pab kho lub hlwb cov paj hlwb thiab txo kev nyuaj siab. Neuroplasticity yog lub hlwb lub peev xwm hloov thiab hloov thaum kawm; nrog rau kev paub zoo los ntawm kev paub thiab kev kawm zoo tuaj.

♦ Kev kawm txog 90 cov neeg mob nrog PTSD tau pom cov txiaj ntsig zoo nrog kev siv Tianeptine hemisulfate monohydrate. Cov kev tshawb fawb kuj pom tau hais tias nrog kev kho mob nrog tianeptine sulfate thiab txo qhov tseem ceeb hauv kev ceeb ntshai. Tianeptine hemisulfate monohydrate muab rau cov neeg mob laus tau pom tias txhim kho txoj kev ntxhov siab vim ua kom tsis muaj zog thiab kev xav li cas.

♦ Cov tsiaj thiab cov tib neeg kev tshawb fawb tau ua los ntawm kev kho mob ntawm Parkinson tus kab mob nrog Tianeptine hemisulfate monohydrate, uas qhia tau cov txiaj ntsig zoo hauv kev txhim kho cov teeb meem kev mob hlwb.

♦ Kev kawm ua ntej ntawm 68 cov kws kho mob nrog ADHD xaus lus tias cov qhab nias ntsuas zoo tuaj yeem zoo tuaj thiab Tianeptine hemisulfate monohydrate zoo rau kev ua kom zoo dua cov peev xwm thiab txo cov kev coj tsis tus.

♦ Tianeptine hemisulfate monohydrate kuj yog ib qho mob zoo (mobkiller), txawm tias cov neeg muaj mob tsis tu ncua. Nws yog ib txoj kev zoo rau kev ua kom muaj cov tsos mob uas muaj feem xyuam nrog plab hnyuv teeb meem thiab.

♦ Lub koom haum ntawm qhov kev soj ntsuam hauv Caracas tau tshawb nrhiav 52-lub limtiam randomized ntawm cov menyuam muaj mob ntsws asthma. Cov neeg mob tau siv Tianeptine hemisulfate monohydrate tsom tus loj nce hauv lub ntsws ua haujlwm.

♦ Txawm tias muaj kev tshawb fawb ntxiv, kev kawm txog 237 tus txiv neej nrog ED tau txiav txim tias tianeptine yuav yog ib qho kev kho zoo.

♦ Tianeptine cov kev mob tshwm sim tsis tuaj yeem cuam tshuam rau acetylcholine lossis ua haujlwm plawv, ua tianeptine ib qho kev xaiv zoo rau cov laus thiab lwm yam


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1 xyuas rau Raw Tianeptine hemisulfate monohydrate hmoov (1224690-84-9)

  1. nyob 5 tawm ntawm 5

    phcoker -

    Tau Raw Tianeptine hemisulfate monohydrate hmoov mus kuaj, kuaj tau qhia tau zoo heev thiab purity!

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